SRL, sarcalumenin, 6345

N. diseases: 77; N. variants: 3
Source: ALL
Disease Score gda Association Type Type Original DB Sentence supporting the association PMID PMID Year
CUI: C0036572
Disease: Seizures
Seizures
0.010 GeneticVariation phenotype BEFREE This work demonstrates that within a chemical series prone to robust M<sub>1</sub> ago-PAM activity, SAR can result, which affords pure M<sub>1</sub> PAMs, devoid of cholinergic toxicity/seizure liability. 30258541 2018